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You are here:Home » Biochemicals » Biochem-Steroids » Eplerenone (CGP 30083, Epoxymexrenone, Inspra, Spiro [9,11-epoxy-9H-cyclopenta[a]phenanthrene-17(2H),2-(3H-furan],pregn-4-ene-7,21-dicarboxylic Acid)

Eplerenone (CGP 30083, Epoxymexrenone, Inspra, Spiro
[9,11-epoxy-9H-cyclopenta[a]phenanthrene-17(2H),2-(3H-furan],pregn-4-ene-7,21-dicarboxyl
ic Acid)

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Specifications

Eplerenone is a potassium-sparing diuretic that selectively blocks aldosterone activation of the mineralcorticoid receptor (IC50=122 nM), demonstrating little activity towards other steroid receptors (IC50 > 9uM for glucocorticoid, androgen, progesterone, and estrogen receptors). Aldosterone antagonists such as this compound have been indicated for the treatment of hypertension and heart failure.
Catalog #E3428-05
Melting Point 225-245°C
Storage and StabilityMay be stored at RT for short-term only. Long-term storage is recommended at -20°C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.
CAS Number107724-20-9
Molecular FormulaC24H30O6
SourceSynthetic
FormWhite to off-white cyrstalline solid
Important NoteThis product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications without the expressed written authorization of United States Biological. Toxicity and Hazards: All products should be handled by qualified personnel only, trained in laboratory procedures.
Alternate namesCGP 30083, Epoxymexrenone, Inspra, Spiro[9,11-epoxy-9H-cyclopenta[a]phenanthrene-17(2H),2?-(3?H-furan],pregn-4-ene-7,21-dicarboxylic Acid, Inspra


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