Technical Data

022861
CAS Number
1232410-49-9
Grade
Highly Purified
MDL Number
MFCD19443686
Molecular Formula
C₁₈H₁₆N₄O₃S
Molecular Weight
368.41
EU Commodity Code
38220090
Shipping Temp
RT
Storage Temp
RT
VE 821
3-amino-6-[4-(methylsulfonyl)phenyl]-N-phenyl-2-pyrazinecarboxamide

VE 821 is a potent and selective inhibitor of DNA damage response kinase, ATR. VE 821 functions to disrupt DNA damage repair system of tumor cells, limiting their abilities for further growth.

Synonyms
3-amino-6-[4-(methylsulfonyl)phenyl]-N-phenyl-2-pyrazinecarboxamide
CAS Number
1232410-49-9
Molecular Formula
C₁₈H₁₆N₄O₃S
Molecular Weight
368.41
Appearance
Supplied as a yellow solid.
Melting Point
247-249°C
Solubility
Chloroform (Slightly), DMSO (Slightly)
Storage and Stability
Store at 4°C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.

Intended for research use only. Not for use in human, therapeutic, or diagnostic applications.

References
1. Finlay, M., et al.: Bioorg. Medn. Chem. Letters., 22, 5352 (2012).
USBio References
No references available
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