Technical Data

256884
CAS Number
896720-20-0
Grade
Highly Purified
Molecular Formula
C24H20Cl2FN5O2
Molecular Weight
500.35
EU Commodity Code
38220090
Shipping Temp
Blue Ice
Storage Temp
4°C
TCS ERK 11e

Potent and selective extracellular signal-related kinase 2 (ERK2) inhibitor (Ki values are <2, 395, 540 and 852 nM for ERK2, GSK-3, Aurora Kinase A and Cdk2 respectively). Potently blocks proliferation of HT29 cells (IC50 = 48 nM). Orally bioavailable.

CAS Number
896720-20-0
Molecular Weight
500.35
Solubility
Soluble to 100 mM in DMSO and to 25 mM in ethanol
Molecular Formula
C24H20Cl2FN5O2
Storage and Stability
Store at 4°C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.

Intended for research use only. Not for use in human, therapeutic, or diagnostic applications.

References
No references available
USBio References
No references available
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